- 第一代: Estranes: Ethisterone
- Etynodiol diacetate
- Lynestrenol
- Norethindrone/Norethisterone
- Norethisterone acetate
- Norethisterone enanthate
- Norethynodrel
- Quingestanol
- 第二代: Estranes: Norethisterone enanthate
- Norgestrienone; Gonanes: 左炔诺孕酮
- Norelgestromin
- Norgestrel
- 第三代: Gonanes: Desogestrel
- Etonogestrel
- Gestodene
- Norgestimate
- 第四代: Estranes: Dienogest; Norpregnanes: Demegestone
- Nomegestrol acetate
- Promegestone
- Trimegestone; Spironolactone derivatives: Drospirenone
- 其他: Pregnanes: Chlormadinone acetate
- 醋酸环丙孕酮
- Medrogestone
- Medroxyprogesterone acetate
- Megestrol acetate; Miscellaneous: 美服培酮
- Ulipristal acetate; Ungrouped: Algestone acetophenide
- Dydrogesterone
- Gestrinone
- 孕酮
- Proligestone